Nrf2及其相关信号通路在膝骨关节炎发病机制中研究
Research progress of Nrf2 and its related signaling pathways in the pathogenesis of knee osteoarthritis
  
DOI:10.3969/j.issn.1006-7108.2025.11.016
中文关键词:  膝骨关节炎  Nrf2信号通路  氧化应激  炎症  铁死亡
英文关键词:knee osteoarthritis  Nrf2 signaling pathway  oxidative stress  inflammation  iron death
基金项目:甘肃省2021年度省级重点人才项目[甘组通字(2021)17号]
作者单位
邵鸿1 赵继荣1* 李喜香2 黄清杰2 陈祁青2 1.甘肃中医药大学甘肃 兰州 730000 2.甘肃省中医院甘肃 兰州 730050 
摘要点击次数: 179
全文下载次数: 0
中文摘要:
      膝骨关节炎(knee osteoarthritis,KOA)是一种以关节软骨退化、软骨下骨改变及滑膜炎症为主要特征,伴随关节疼痛和功能障碍的慢性退行性关节疾病。核转录因子红系2相关因子2(Nrf2)是细胞内的重要抗氧化调节因子,其通过调控下游抗氧化、抗炎和抗铁死亡基因的表达,在维持细胞氧化还原平衡和保护组织功能方面发挥关键作用。研究表明,Nrf2信号通路通过多种机制在KOA的发病中发挥保护作用,Nrf2激活后通过上调HO-1、NQO1、SOD等抗氧化酶的表达,减少ROS积累,缓解氧化应激,保护软骨细胞免受氧化损伤;Nrf2通过抑制NF-κB和NLRP3炎症小体的激活,减少促炎性因子(如IL-1β、TNF-α)的产生,减轻滑膜炎症和软骨退化;此外,Nrf2通过调节GPX4表达,抑制脂质过氧化和铁死亡,保护软骨细胞,进一步延缓KOA进展。该综述系统总结了Nrf2信号通路在KOA中抗氧化、抗炎和抗铁死亡具体机制,探讨其在KOA中的核心作用及治疗潜力,强调这些机制单独或相互作用对KOA的影响,为理解KOA的发病机制提供了新视角,为开发针对KOA的多靶点干预策略和高效治疗方法提供了理论依据与研究方向。
英文摘要:
      Knee osteoarthritis (KOA) is a chronic degenerative joint disease characterized by articular cartilage degeneration, subchondral bone changes, and synovial inflammation, accompanied by joint pain and dysfunction. Nrf2 (nuclear factor erythroid 2-related factor 2) is an important antioxidant regulator in cells. It plays a key role in maintaining cell redox balance and protecting tissue function by regulating the expression of downstream antioxidant, anti-inflammatory, and anti-ferroptosis genes. Studies have shown that Nrf2 signaling pathway plays a protective role in the pathogenesis of KOA through a variety of mechanisms. After activation of Nrf2, it can reduce ROS accumulation, alleviate oxidative stress, and protect chondrocytes from oxidative damage by up-regulating the expression of antioxidant enzymes such as HO-1, NQO1, and SOD. Nrf2 attenuates synovial inflammation and cartilage degeneration by inhibiting the activation of NF-κB and NLRP3 inflammasome, reducing the production of pro-inflammatory factors (such as IL-1β, TNF-α). In addition, Nrf2 protects chondrocytes by regulating GPX4 expression, inhibiting lipid peroxidation and ferroptosis, and further delaying KOA. This review systematically summarizes the specific mechanisms of Nrf2 signaling pathway in anti-oxidation, anti-inflammatory, and anti-ferroptosis in KOA, discusses its core role and therapeutic potential in KOA, and emphasizes the effects of these mechanisms alone or in interaction on KOA. It provides a new perspective for understanding the pathogenesis of KOA, and provides a theoretical basis and research direction for the development of multi-target intervention strategies and efficient treatment methods for KOA.
查看全文  查看/发表评论  下载PDF阅读器
关闭
function PdfOpen(url){ var win="toolbar=no,location=no,directories=no,status=yes,menubar=yes,scrollbars=yes,resizable=yes"; window.open(url,"",win); } function openWin(url,w,h){ var win="toolbar=no,location=no,directories=no,status=no,menubar=no,scrollbars=yes,resizable=no,width=" + w + ",height=" + h; controlWindow=window.open(url,"",win); } &et=FC9DA7BF2F842A3BAE24B54F70914FE6B1CB3199CBE13495B9E7ADCC476C958092A36FEE0E4023B21C0A439A4FA94C26A131EA8D51D4C5964EA44A2E08E94D444BC51A46A8FA5D97DE6E5AB680D890B4433ED0B67434C2761F1FF9D06E3BBF597DE9D75DFA5C804F&pcid=A9DB1C13C87CE289EA38239A9433C9DC&cid=527A01A248DACB72&jid=CA678592D11E309E8E3FB3B2BFE9BE1A&yid=E6A891D2134F30C0&aid=&vid=&iid=708DD6B15D2464E8&sid=4F4D699E68EBCB79&eid=00B387A522283F93&fileno=202511016&flag=1&is_more=0"> var my_pcid="A9DB1C13C87CE289EA38239A9433C9DC"; var my_cid="527A01A248DACB72"; var my_jid="CA678592D11E309E8E3FB3B2BFE9BE1A"; var my_yid="E6A891D2134F30C0"; var my_aid="";