六味地黄丸调控SLC31A1/FDX1轴抑制铜死亡改善糖尿病性骨质疏松的作用及机制
The effect and mechanism of Liuwei Dihuang pill in regulating the SLC31A1/FDX1 axis, inhibiting cuproptosis, and relieving diabetic osteoporosis
  
DOI:10.3969/j.issn.1006-7108.2026.01.003
中文关键词:  糖尿病性骨质疏松  铜死亡  铜稳态  六味地黄丸
英文关键词:diabetic osteoporosis  cuproptosis  copper homeostasis  Liuwei Dihuang pill
基金项目:广东省自然科学基金(2021A1515010725)
作者单位
连勇1 谢志兴1 陆嘉欣1 潘兆丰1 陈庆真2 邵敏2* 1.广州中医药大学第三临床医学院广东 广州 510405 2.广州中医药大学第三附属医院广东 广州 510405 
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中文摘要:
      目的 探讨六味地黄丸对SLC31A1/FDX1轴的调控作用及其对糖尿病性骨质疏松症(diabetic osteoporosis,DOP)的防治机制。方法 临床研究:采集DOP组、骨质疏松(osteoporosis,OP)组及对照组(Control)受试者的血清和骨组织样本,检测其血清铜离子含量、铜蓝蛋白(ceruloplasmin,Cp)水平及骨组织内铜离子含量,分析铜稳态与DOP的关系;动物实验:80只小鼠随机分为空白组、模型组、低剂量六味地黄丸组和高剂量六味地黄丸组,干预8周后,观察六味地黄丸对小鼠血糖、体重、饮食量、尿量的影响;Elabscience络合法检测小鼠血清及骨组织内铜含量;Micro-CT检测骨微细结构(BV/TV、Tb.Th、Tb.N)变化;苏木精-伊红(H&E)和免疫组化(IHC)检测骨组织形态学变化;Western blot技术检测铜死亡相关蛋白(PDHA1、DLD、DLAT)及SLC31A1/FDX1轴表达水平。结果 临床研究:糖尿病性骨质疏松组血清和骨组织中的铜离子含量及铜蓝蛋白水平显著高于骨质疏松组和对照组,提示铜稳态异常与DOP的发生密切相关。动物实验:六味地黄丸显著降低了糖尿病骨质疏松小鼠的血糖水平,改善了骨微细结构,减少了骨组织内铜含量,并上调了铜死亡相关蛋白FDX1的表达,下调了铜转运酶SLC31A1的表达。结论 铜死亡机制参与了糖尿病性骨质疏松的发病过程。六味地黄丸通过调控SLC31A1/FDX1轴,抑制铜死亡过程,改善骨微细结构和骨组织形态,从而发挥防治糖尿病性骨质疏松的作用。
英文摘要:
      Objective To verify the role of cuproptosis in the pathogenesis of diabetic osteoporosis (DOP) and to explore the mechanism by which Liuwei Dihuang pill regulates the SLC31A1/FDX1 axis and its protective effects on DOP. Methods Clinical research: Blood samples from DOP, osteoporosis (OP), and control patients were collected to detect serum copper levels, copper ceruloplasmin (Cp) levels, and bone tissue copper content. The relationship between copper homeostasis and DOP was analyzed Animal experiments: In this study, eighty mice were randomly divided into four groups: control group, model group, low-dose herbal formulation group, and high-dose herbal formulation group. After an 8-week intervention, the effects of the herbal formulation on blood glucose, body weight, food intake, and urine output in the mice were observed. Copper levels in mouse serum and bone tissue were detected using Elabscience legal method. Bone microstructure (BV/TV,Tb.Th,Tb.N) was examined using micro-CT. Bone structural changes were assessed using hematoxylin and Eosin staining and immunohistochemistry. Western blotting was used for the expression levels of cuproptosis-related proteins (PDHA1, DLD, DLAT) and the SLC31A1/FDX1 axis. Results Clinical research: Serum and bone tissue copper levels, as well as copper ceruloplasmin levels, were significantly higher in diabetic bone quality deficiency patients than in osteoporosis patients and healthy controls, suggesting a close relationship between copper metabolism and DOP. Animal experiments: Liuwei Dihuang pill effectively inhibited copper-induced apoptosis, improved bone microstructure and bone tissue organization, thereby exerting protective effects against diabetic bone quality deficiency. Conclusion Liuwei Dihuang pill regulates the SLC31A1/FDX1 axis by inhibiting cuproptosis, thereby improving bone microstructure and bone tissue organization, ultimately achieving its therapeutic effect on diabetic bone quality deficiency.
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